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purity 99% Pikamilon / Picamilon Sodium Salt Powder, nutritional pikamilone CAS 62936-56-5, 34562-97-5
Chemical Information:
CAS Number: 62936-56-5
Purity: ≥98%
Molecular Weight: 230.20 g/mol
Melting Point: 208.0-212.0°C
Molecular Formula: C10H11N2O3 •Na
Synonyms: Picamilon, Pikamilone sodium salt, Pikamilone, Pikamilon sodium salt, Nicotinoyl-GABA sodium salt, 4-(Pyridine-3-carbonylamino)butanoic acid sodium salt, Monosodium 4-(pyridine-3-carbonylamino)butanoate, Monosodium 4-Nicotinoylaminobutyrate, N-(3-Pyridinylcarbonyl)-4-aminobutyric acid sodium
PubChem CID: 23663986
SMILES: C1=CC(=CN=C1)C(=O)NCCCC(=O)[O-].[Na+]
| Product Name |
Pikamilone |
| Batch No. |
14121501 |
Mfg. date |
2014-12-15 |
| Test Date |
2014-12-25 |
Exp. date |
2016-12-14 |
| Tests |
Specifications |
Results |
| Description |
White to yellowish powder, very hygroscopic. |
Off-white powder, very hygroscopic. |
| Solubility |
Freetly soluble In water and methanol and dichloromethane |
Complies |
| Identification |
(1)By IR, To match with working standard |
Complies |
| (2)It gives reaction of sodium |
Complies |
| Impurities A |
≤0.1% |
Not detected |
| Related compounds |
Any impurity ≤0.1% |
<0.1% |
| Total impurities ≤0.4% |
0.25% |
| Residual Solvents |
Acetidin≤ 0.5% |
Not detected |
| Dichloromethane≤ 0.06% |
Not detected |
| Methanol≤ 0.3% |
Not detected |
| Acetone ≤ 0.5% |
Not detected |
| Acetonitrile≤0.041% |
Not detected |
| Ethanol≤0.5% |
0.04% |
| N, N-dimethylformamide≤0.088% |
Not detected |
| Water |
≤ 5.0% |
1.38% |
| Assay |
99.0%-101.0%(On anhydrous basis) |
99.98% |
| Conclusion |
Conform to EP8.0 |
Technical Information:
Application: Picamilon is a linked derivative of the vitamin Niacin (vitamin B3, nicotinic acid) with the inhibitory neurotransmitter GABA, useful in the research of BBB penetrant molecules which hydrolyse to yield GABA.
Appearance: White or off-white powder
Physical State: Solid
Solubility: Freely soluble in Ethanol, Water.
Storage: Store at room temperature or cooler, in a sealed airtight container, protected from heat, light and humidity.
Stability: Stable for at least two years when stored as above.
Biochemical Activity:
Picamilon is a amide derivative of the vitamin Niacin (vitamin B3, nicotinic acid) and the inhibitory neurotransmitter GABA. It was developed in the Soviet Union in 1969 and further studied in both Russia and Japan as a prodrug of GABA.
